CB2 receptor antagonist 2
CB2 receptor antagonist 2 (compound 39) is a potent antagonist of CB2 with an IC50 value of 0.33 μM. CB2 receptor antagonist 2 has strong interactions with L17, W6.48, V6.51, and C7.42[1].
Product Specifications
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/cb2-receptor-antagonist-2.html
Solubility
10 mM in DMSO
Smiles
CCCS(=O)(OC1=CC(/C=C(SC(N2C(C)C)=O)/C2=O)=CC=C1OC)=O
Molecular Formula
C17H21NO6S2
Molecular Weight
399.48
References & Citations
[1]Yu-Chieh Wu, et al. Novel 4-aminoquinoline analogs targeting the HIF-1α signaling pathway. Future Med Chem. 2023,15,17.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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