D4R agonist-1

D4R agonist-1 (Compound 16f) is a D4R partial agonist (Ki: 2.2 nM) . D4R agonist-1 is metabolically stable in rat and human liver microsomes. D4R agonist-1 can be used for research of neuropsychiatric disorders[1].

Product Specifications

CAS Number

[2826198-44-9]

UNSPSC

12352005

Target

Dopamine Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/d4r-agonist-1.html

Solubility

10 mM in DMSO

Smiles

C12=CC=CC=C1N=C(S2)CCCN3CCN(CC3)C4=NC=CC=C4

Molecular Formula

C19H22N4S

Molecular Weight

338.47

References & Citations

[1]Boateng CA, et al. Pharmacology and Therapeutic Potential of Benzothiazole Analogues for Cocaine Use Disorder. J Med Chem. 2023 Aug 30.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Available Sizes

Curated Selection

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