PLK1-IN-5
PLK1-IN-5 is a potent PLK1 inhibitor with an IC50 of [1].
Product Specifications
CAS Number
1001343-34-5
UNSPSC
12352005
Target
Polo-like Kinase (PLK)
Type
Reference compound
Related Pathways
Cell Cycle/DNA Damage
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/plk1-in-5.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=CC=C(C(OC)=C1)NC2=NC=C3C(N(C4CCCC4)C(CC(N3C)=O)C)=N2)NC5CCN(CC5)C
Molecular Formula
C28H39N7O3
Molecular Weight
521.65
References & Citations
[1]Jianping Cai, et al. Substituted pyrimidodiazepines useful as plk1 inhibitors. WO2008113711A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
PLK1
Frequently Asked Questions
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