TRPV1 activator-1
TRPV1 activator-1 (compound 8), a capsaicin analog, has an altered neck structure. TRPV1 activator-1 interacts specifically with T551 residue[1].
Product Specifications
CAS Number
1803181-80-7
UNSPSC
12352005
Target
TRP Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/trpv1-activator-1.html
Solubility
10 mM in DMSO
Smiles
CC(C)/C=C/CCCCC(NCC1=CC=C(O)C(OC)=C1)=S
Molecular Formula
C18H27NO2S
Molecular Weight
321.48
References & Citations
[1]Fan Yang, et al. Structural mechanism underlying capsaicin binding and activation of the TRPV1 ion channel. Nat Chem Biol. 2015 Jul;11 (7) :518-524.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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