β2AR/M3-receptor agonist-1

β2AR/M3-receptor agonist-1 (example 9) is a potent β2AR and M3 receptor agonist. β2AR/M3-receptor agonist-1 shows M3 receptor affinity with a pIC50 value of 9.3. β2AR/M3-receptor agonist-1 has the potential for the research of respiratory tract disorders[1].

Product Specifications

CAS Number

[1206887-00-4]

UNSPSC

12352005

Target

Adrenergic Receptor; mAChR

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Metabolism-sugar/lipid metabolism

Field of Research

Metabolic Disease

Assay Protocol

https://www.medchemexpress.com/β2ar-m3-receptor-agonist-1.html

Solubility

10 mM in DMSO

Smiles

O=CO.O=C1NC2=C(OC1)C(C(CNCCC3=CC=C(C=C3)OCCCNCC4=CC(C(C5=CC=CC=C5)(C6=CC=CC=C6)O)=NO4)O)=CC=C2O.[x]

Molecular Formula

C38H40N4O7.xCH2O2

References & Citations

[1]Jonathan Mark Sutton, et al. Nitrogen containing heterocyclic compounds useful as bifunctional modulators of m3 receptors and beta-2 receptors. WO2010015792A1.