Mrgx2 antagonist-2
Mrgx2 antagonist-2 is a Mrgx2 antagonist (Example 123 in reference patent) with a pIC50 of 8.6. Mrgx2 antagonist-2 can be used in the research of MrgX2 -mediated diseases or disorders[1].
Product Specifications
CAS Number
[2767111-67-9]
UNSPSC
12352005
Target
Mas-related G-protein-coupled Receptor (MRGPR)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
COVID-19-immunoregulation
Field of Research
Cancer; Inflammation/Immunology; Neurological Disease
Assay Protocol
https://www.medchemexpress.com/mrgx2-antagonist-2.html
Solubility
10 mM in DMSO
Smiles
FC1([C@@H](C2=CC=[N+]([O-])C=C2)CN(CC1)[C@@H](C)C(NC3=NC=C(OC4=C(C=C(C=C4)F)F)N=C3)=O)F
Molecular Formula
C23H21F4N5O3
Molecular Weight
491.44
References & Citations
[1]Edward Brnardic, et al. Mrgx2 antagonists. Patent. WO2022073904.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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