DC-CPin7
DC-CPin7 is a potent inhibitor of CREB-binding protein (CBP) bromodomain with an IC50 of 2.5 μM[1].
Product Specifications
CAS Number
893781-17-4
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/dc-cpin7.html
Solubility
10 mM in DMSO
Smiles
OC(C1C(CC=CC1)C(NC2=CC3=C(C=C2)N(C(OC)=O)CCC3)=O)=O
Molecular Formula
C19H22N2O5
Molecular Weight
358.39
References & Citations
[1]Chen Y, et al. Design, synthesis, and biological evaluation of tetrahydroquinolin derivatives as potent inhibitors of CBP bromodomain. Bioorg Chem. 2020 Aug;101:103991.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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