5-HT7 receptor ligand 1
5-HT7 receptor ligand 1 (Compound 5c) is a 5-HT7 receptor ligand with a Ki of 8 nM. 5-HT7 receptor ligand 1 is not hepatotoxic and exhibit moderate potential interaction with other agents metabolized by CYP3A4 or CYP2D6[1].
Product Specifications
CAS Number
2758571-64-9
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/5-ht7-receptor-ligand-1.html
Solubility
10 mM in DMSO
Smiles
NC1=NC(NCCC2=CNC3=C2C=CC=C3)=NC(NCCC4=CC=CC=C4)=N1
Molecular Formula
C21H23N7
Molecular Weight
373.45
References & Citations
[1]Kułaga D, et al. Aminotriazines with indole motif as novel, 5-HT7 receptor ligands with atypical binding mode. Bioorg Chem. 2020 Nov;104:104254.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT7 Receptor; MUC3
Frequently Asked Questions
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