CB2 receptor antagonist 1
Hexyl resorcinol derivative 29 has been proved to be a CB2 selective competitive antagonist / reverse agonist with good potency. Olivanol and 5- (2-methyloctane-2-yl) resorcinol derivatives 23 and 24 showed significant antinociceptive activity. Compound 24 was shown to activate cannabinoid and TRPV1 receptors.
Product Specifications
CAS Number
2772693-05-5
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/cb2-receptor-antagonist-1.html
Solubility
10 mM in DMSO
Smiles
CCCCCCC1=CC=C(C=C1OC)OCCCCCCCCCCC(NCC2CC2)=O
Molecular Formula
C28H47NO3
Molecular Weight
445.68
References & Citations
[1]Brizzi A, et al. Synthetic bioactive olivetol-related amides: The influence of the phenolic group in cannabinoid receptor activity. Bioorg Med Chem. 2020 Jun 1;28 (11) :115513.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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