BET-IN-10
BET-IN-10 is a BET inhibitor with anticancer effects. BET-IN-10 inhibits the cell growth of MV4-11 cells with an IC50 of 26.5 nM (WO2022012456A1; example 6) [1].
Product Specifications
CAS Number
2758778-95-7
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/bet-in-10.html
Solubility
10 mM in DMSO
Smiles
CCNC(C1=CC2=C(C(N(C=C2C3=C(C=C(S3)C(C)(O)C)OC4=C(C=C(C=C4C)F)C)C)=O)N1)=O
Molecular Formula
C26H28FN3O4S
Molecular Weight
497.58
References & Citations
[1]Haiquan Fang, et al. Novel heterocyclic compounds as bet inhibitors. WO2022012456A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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