CB1R Allosteric modulator 2
CB1R Allosteric modulator 2 (compound 18) is a potent CB1R allosteric modulator. CB1R Allosteric modulator 2 shows negatively affects the functional activity of orthosteric ligands (NAM) at CB1Rs[1].
Product Specifications
CAS Number
2513102-64-0
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/cb1r-allosteric-modulator-2.html
Solubility
10 mM in DMSO
Smiles
O=C(NC1=CC(NC2=CC=C(C=C2)F)=CC=C1)NC3=CC=C(C=C3)Cl
Molecular Formula
C19H15ClFN3O
Molecular Weight
355.79
References & Citations
[1]Meini S, et al. PSNCBAM-1 analogs: Structural evolutions and allosteric properties at cannabinoid CB1 receptor. Eur J Med Chem. 2020 Oct 1;203:112606.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CB1
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