CB1R Allosteric modulator 1
CB1R Allosteric modulator 1 (compound 11) is a potent CB1R allosteric modulator. CB1R Allosteric modulator 1 shows negatively affects the functional activity of orthosteric ligands (NAM) at CB1Rs[1].
Product Specifications
CAS Number
2513102-41-3
UNSPSC
12352005
Target
Cannabinoid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/cb1r-allosteric-modulator-1.html
Solubility
10 mM in DMSO
Smiles
O=C(NC1=CC(C2=CC=CC(N3CCCCC3)=C2)=CC=C1)NC4=CC=C(C=C4)Cl
Molecular Formula
C24H24ClN3O
Molecular Weight
405.92
References & Citations
[1]Meini S, et al. PSNCBAM-1 analogs: Structural evolutions and allosteric properties at cannabinoid CB1 receptor. Eur J Med Chem. 2020 Oct 1;203:112606.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
CB1
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