CB2R probe 1

CB2R probe 1 is a safe and green CB2R (cannabinoid 2 receptor) fluorescent probe with an Ki of 130 nM. CB2R probe 1 shows low cytotoxicity in cancer cells[1].

Product Specifications

CAS Number

[2634714-79-5]

UNSPSC

12352005

Target

Cannabinoid Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Cancer-programmed cell death

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/cb2r-probe-1.html

Solubility

10 mM in DMSO

Smiles

CN(C1=CC2=C(C(N(C2=O)CCCCCCN3C=C(C(C4=CC=CC=C43)=O)C(N[C@@]5(CC6C7)CC7CC(C6)C5)=O)=O)C=C1)C

Molecular Formula

C36H42N4O4

Molecular Weight

594.74

References & Citations

[1]Spinelli F, et al. Design and synthesis of fluorescent ligands for the detection of cannabinoid type 2 receptor (CB2R) . Eur J Med Chem. 2020 Feb 15;188:112037.