Bromodomain inhibitor-9
Bromodomain inhibitor-9 is a Bromodomains inhibitor that selectively inhibits BRD4-1 (Kd: 12 nM) . Bromodomain inhibitor-9 can be used in the research of diseases or conditions associated with systemic or tissue inflammation, lipid metabolism, fibrosis or chronic autoimmune diseases[1].
Product Specifications
CAS Number
[1870849-34-5]
UNSPSC
12352005
Hazard Statement
H315-H319-H320
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Metabolism-sugar/lipid metabolism
Field of Research
Metabolic Disease; Inflammation/Immunology
Assay Protocol
https://www.medchemexpress.com/bromodomain-inhibitor-9.html
Solubility
10 mM in DMSO
Smiles
O=C1C=C(C)C2=C(N1)C=C(C)C(NC(C3=CC(S(=O)(N(C)C)=O)=CC=C3N4CCOCC4)=O)=C2
Molecular Formula
C24H28N4O5S
Molecular Weight
484.57
Precautions
P264-P280-P302+P352-P305+P351+P338-P362
References & Citations
[1]Gerner Seitzberg, et al. Heterocyclic compounds as inhibitors of bromodomains and their preparation. Patent WO2016016316.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
BRD4
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