SGC-AAK1-1N
SGC-AAK1-1N is a potent and selective AAK1 (AP2 associated kinase 1) inhibitor, with an IC50 of 1.8 μM[1].
Product Specifications
CAS Number
[2242913-80-8]
UNSPSC
12352005
Target
AAK1
Type
Reference compound
Related Pathways
Neuronal Signaling
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/sgc-aak1-1n.html
Purity
97.9
Solubility
10 mM in DMSO
Smiles
CC(C(NC1=NNC2=C1C=CC(C3=CC(NS(=O)(C4CC4)=O)=CC=C3)=C2)=O)C
Molecular Formula
C20H22N4O3S
Molecular Weight
398.48
References & Citations
[1]Wells C, et al. SGC-AAK1-1: A Chemical Probe Targeting AAK1 and BMP2K. ACS Med Chem Lett. 2019 Oct 23;11 (3) :340-345.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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