BET bromodomain inhibitor 2
BET bromodomain inhibitor 2 is a potent BET bromodomain inhibitor with an IC50 of 14.1 µM[1].
Product Specifications
CAS Number
2414195-69-8
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/bet-bromodomain-inhibitor-2.html
Solubility
10 mM in DMSO
Smiles
CCN(S(=O)(C1=CC=C(C(C2=CC(OC)=C(C=C2)OC)=C1)[C@H]3CC(N(C3)C)=O)=O)CC
Molecular Formula
C23H30N2O5S
Molecular Weight
446.56
References & Citations
[1]J P Hilton-Proctor, et al. Substituted 1-methyl-4-phenylpyrrolidin-2-ones - Fragment-based design of N-methylpyrrolidone-derived bromodomain inhibitors. Eur J Med Chem. 2020 Apr 1;191:112120.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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