KCa1.1 channel activator-2
KCa1.1 channel activator-2 (compound 3F), a Quercetin hybrid derivative, is a selective vascular KCa1.1 channel stimulator. KCa1.1 channel activator-2 exhibits potent myorelaxant activity[1].
Product Specifications
UNSPSC
12352005
Target
Potassium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/kca1-1-channel-activator-2.html
Solubility
10 mM in DMSO
Smiles
O=C(OC1=CC2=C(C(O)=C1)C(C(O)=C(O2)C3=CC=C(C(O)=C3)O)=O)CCCCC4CCSS4
Molecular Formula
C23H22O8S2
Molecular Weight
490.55
References & Citations
[1]Carullo G, et, al. Design, synthesis and pharmacological evaluation of ester-based quercetin derivatives as selective vascular K Ca 1.1 channel stimulators. Bioorg Chem. 2020 Dec;105:104404.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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