MC2652
MC2652 (compound 1a) is a potent LSD1 inhibitor. MC2652 displays high inhibiting effects in MV4-11 and NB4 leukaemia cells. MC2652 shows antiproliferative activity against prostate cancer LNCaP cells[1].
Product Specifications
CAS Number
2771425-46-6
UNSPSC
12352005
Target
Histone Demethylase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/mc2652.html
Solubility
10 mM in DMSO
Smiles
NC1CC1C2=CC=C(C=C2)NC(C3=CC=C(C=C3)C4=CC=CC=C4)=O
Molecular Formula
C22H20N2O
Molecular Weight
328.41
References & Citations
[1]Fioravanti R, et al. Heterocycle-containing tranylcypromine derivatives endowed with high anti-LSD1 activity. J Enzyme Inhib Med Chem. 2022 Dec;37 (1) :973-985.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
KDM1/LSD1
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