RSK-IN-1
RSK-IN-1 (compound 7d) is a RSK inhibitor that inhibits the YB-1 phosphorylation. RSK-IN-1 has anti-tumor effects[1].
Product Specifications
CAS Number
2761698-77-3
UNSPSC
12352005
Target
Ribosomal S6 Kinase (RSK) ; YB-1
Type
Reference compound
Related Pathways
Cell Cycle/DNA Damage; MAPK/ERK Pathway
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/rsk-in-1.html
Solubility
10 mM in DMSO
Smiles
CC1=C2C=CC=CC2=C(C=C1)C3=CC=NC=C3C4=CC=C(C(O)=C4)O
Molecular Formula
C22H17NO2
Molecular Weight
327.38
References & Citations
[1]Yi-Man Cui, et al. Design, synthesis and anti-breast cancer evaluation of biaryl pyridine analogues as potent RSK inhibitors. Bioorg Med Chem Lett. 2022 Mar 1;59:128565.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog