BRD4-BD1-IN-1
BRD4-BD1-IN-1 (Compound 9a) is a BRD4-BD1 inhibitor with an IC50 of 38.20 μM[1].
Product Specifications
CAS Number
2761321-18-8
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/brd4-bd1-in-1.html
Solubility
10 mM in DMSO
Smiles
CC(OCC1=NC2=C(N1CC3=CC(Br)=CC=C3)C(NC(N2C)=O)=O)=O
Molecular Formula
C16H15BrN4O4
Molecular Weight
407.22
References & Citations
[1]Chang Y, et al. Design, synthesis, biological evaluation, and molecular docking of 1, 7-dibenzyl-substituted theophylline derivatives as novel BRD4-BD1-selective inhibitors. Medicinal Chemistry Research, 2021, 30 (8) : 1453-1468.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
BRD4
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