ER degrader 1
ER degrader 1 is a potent degrader of estrogen receptor (ER) . The estrogen signaling system plays an important role in regulating cell growth, differentiation and apoptosis. ER degrader 1 has the potential for the research of cancer diseases (extracted from patent WO2021139756A1, compound 11) [1].
Product Specifications
CAS Number
2667015-33-8
UNSPSC
12352005
Target
Estrogen Receptor/ERR
Type
Reference compound
Related Pathways
Vitamin D Related/Nuclear Receptor
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/er-degrader-1.html
Solubility
10 mM in DMSO
Smiles
OCC(F)(F)CN1[C@@](C2=C(C=C(C=N2)N[C@@H]3CN(CC3)CCCF)F)([H])C4=C(C[C@H]1C)C=C5C(OCO5)=C4
Molecular Formula
C26H32F4N4O3
Molecular Weight
524.55
References & Citations
[1]Fanglong Yang, et al. Tricyclic tetrahydroisoquinoline derivatives, their preparation methods and their application in medicine. Patent WO2021139756A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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