BRD4-BD1/2-IN-2
BRD4-BD1/2-IN-2 is a potent BRD4 BD2 inhibitor with IC50s of [1].
Product Specifications
CAS Number
[2743464-27-7]
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/brd4-bd1-2-in-2.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=CC(C(C2=CC3=NN(CC(C)(C)O)C=C3C=C2OC4=C(C)C=CC=C4C)=CN5C)=C(N1)C5=O)NCC
Molecular Formula
C30H33N5O4
Molecular Weight
527.61
References & Citations
[1]Compound functioning as bromodomain protein inhibitor, and composition. WO2021233371A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
043992-ML650 100 µL
ZBTB12, CT (ZBTB12, C6orf46, G10, NG35, Zinc finger and BTB domain-containing protein 12, Protein G10) (MaxLight 650) discontinued
Ask
View Details 