BRD4-BD1/2-IN-1
BRD4-BD1/2-IN-1 is a potent BRD4 inhibitor with IC50s of [1].
Product Specifications
CAS Number
[1781219-19-9]
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/brd4-bd1-2-in-1.html
Solubility
10 mM in DMSO
Smiles
O=C1C2=C(C(C3=CC4=C(C=C3OC5=CC=C(C=C5F)F)N=CN4)=CN1C)C=CN2
Molecular Formula
C21H14F2N4O2
Molecular Weight
392.36
References & Citations
[1]Bicyclic heterocycles as bet protein inhibitors. US20150148375A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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