ERK1/2 inhibitor 8
ERK1/2 inhibitor 8 is a potent ERK inhibitor with an IC50 of 0.48 nM for ERK2 (WO2021110168A1, WX007) [1].
Product Specifications
CAS Number
2648368-43-6
UNSPSC
12352005
Target
ERK
Type
Reference compound
Related Pathways
MAPK/ERK Pathway; Stem Cell/Wnt
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/erk1-2-inhibitor-8.html
Solubility
10 mM in DMSO
Smiles
O=C1C2=C(C3(COC3)N1CC4=CC(Cl)=CC=C4)SC(C5=C(C)C=NC(NC6=CC=NN6C)=N5)=N2
Molecular Formula
C23H20ClN7O2S
Molecular Weight
493.97
References & Citations
[1]WO2021110168A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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