S1P2 antagonist 1
S1P2 antagonist 1 is an orally bioavailable S1P2 antagonist against fibrotic diseases.
Product Specifications
CAS Number
2262402-83-3
UNSPSC
12352005
Target
LPL Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/s1p2-antagonist-1.html
Solubility
10 mM in DMSO
Smiles
OC([C@@H](C)N1N=C(CN2N=C(C=C(Cl)C(OCC3CC3)=C4)C4=C2)C5=CC=CC=C5C1=O)=O
Molecular Formula
C23H21ClN4O4
Molecular Weight
452.89
References & Citations
[1]Mammoliti O, et al. Discovery and Optimization of Orally Bioavailable Phthalazone and Cinnolone Carboxylic Acid Derivatives as S1P2 Antagonists against Fibrotic Diseases. J Med Chem. 2021 Oct 14;64 (19) :14557-14586.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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