HA3AR agonist 1

HA3AR agonist 1 is a potent human A3 adenosine receptor (hA3AR) agonist with a Ki value of 2.40 nM.

Product Specifications

CAS Number

[2821704-65-6]

UNSPSC

12352005

Target

Adenosine Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein

Applications

Neuroscience-Neuromodulation

Field of Research

Others

Assay Protocol

https://www.medchemexpress.com/ha3ar-agonist-1.html

Solubility

10 mM in DMSO

Smiles

O[C@H]1[C@H](N2C=NC3=C(NC)N=CN=C23)SC[C@H]1N

Molecular Formula

C10H14N6OS

Molecular Weight

266.32

References & Citations

[1]Lee Y, et al. Subtle Chemical Changes Cross the Boundary between Agonist and Antagonist: New A3 Adenosine Receptor Homology Models and Structural Network Analysis Can Predict This Boundary. J Med Chem. 2021 Sep 9;64 (17) :12525-12536.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

Adenosine A3 receptor (A3R)

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