AHR antagonist 5 (hemimaleate)
AHR antagonist 5 hemimaleate, a potent and orally active aryl hydrocarbon receptor (AHR) antagonist, has an IC50 of [1].
Product Specifications
UNSPSC
12352005
Target
Aryl Hydrocarbon Receptor
Type
Reference compound
Related Pathways
Immunology/Inflammation
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ahr-antagonist-5-hemimaleate.html
Solubility
10 mM in DMSO
Smiles
CC(C1=C2N(N=C1)C(N[C@H]3CC(C4=CC=CC=C4N5)=C5CC3)=NC(C6=CN=CC(F)=C6)=N2)C.O=C(O)/C=C\C(O)=O.[1/2]
Molecular Formula
C27H26O2FN7
Molecular Weight
499.55
References & Citations
[1]Alfredo C. Castro, et al. Indole ahr inhibitors and uses thereof. WO2018195397A2.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Phase 1
Frequently Asked Questions
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