MCHR1 antagonist 3
MCHR1 antagonist 3 is a potent the melanin-concentrating hormone receptor-1 (MCHR1) antagonist. MCHR1 antagonist 3 is used to regulate energy metabolism[1].
Product Specifications
CAS Number
[1069622-60-1]
UNSPSC
12352005
Target
MCHR1 (GPR24)
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Endocrinology; Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/mchr1-antagonist-3.html
Solubility
10 mM in DMSO
Smiles
O=C(N1C2CC3=C(C=CC=C3)C2)N(CC)C4(CCN(CC5=CC=C(N6CCCC6)C=C5)CC4)C1=O
Molecular Formula
C29H36N4O2
Molecular Weight
472.62
References & Citations
[1]Rowbottom MW, et al. Synthesis and structure-activity relationships of spirohydantoin-derived small-moleculeantagonists of the melanin-concentrating hormone receptor-1 (MCH-R1) . Bioorg Med Chem Lett. 2007 Apr 15;17 (8) :2171-8.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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