CPI-1328
Product Specifications
UNSPSC Description
CPI-1328 is an EZH2 inhibitor with a Ki value of 63 fM.
Target Antigen
Histone Methyltransferase
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/cpi-1328.html
Solubility
10 mM in DMSO
Smiles
ClC1=C2C(O[C@](O2)([C@]3([H])CC[C@H](CC3)N(C)C)C)=C(C4=C1CCN(C4=O)CC5=C(C=C(NC5=O)C)SC)C
Molecular Weight
546.12
References & Citations
[1]Stuckey JI, et al. Identification and characterization of second-generation EZH2 inhibitors with extended residence times and improved biological activity. J Biol Chem. 2021 Jan-Jun;296:100349.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-134899/CPI-1328-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-134899/
Clinical Information
No Development Reported
CAS Number
2390367-27-6
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
![Mouse Monoclonal Cytochrome P450 4A Antibody (M25-P2A10) [DyLight 488]](https://cdn.genprice.uk/genprice/genprice2.png)
NBP2-50212G 0.1 mL
Mouse Monoclonal Cytochrome P450 4A Antibody (M25-P2A10) [DyLight 488]
Ask
View Details 