Pilsicainide
Pilsicainide (SUN 1165 free acid) is a potent sodium channel blocker and potent class Ic antiarrhythmic agent[1][2].
Product Specifications
CAS Number
[88069-67-4]
Product Name Alternative
SUN 1165 (free base) ; Pilzicainide
UNSPSC
12352005
Hazard Statement
H302-H315-H319-H335
Target
Sodium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/pilsicainide.html
Solubility
10 mM in DMSO
Smiles
O=C(NC1=C(C)C=CC=C1C)CC23CCCN2CCC3
Molecular Formula
C17H24N2O
Molecular Weight
272.39
Precautions
P261-P264-P270-P271-P280-P302+P352-P304+P340-P305+P351+P338-P330-P362+P364-P403+P233-P405-P501
References & Citations
[1]Yamakawa M, et al. Effect of sodium channel blocker, pilsicainide hydrochloride, on net inward current of atrial myocytes in thyroid hormone toxicosis rats. Thyroid. 2005 Jul;15 (7) :653-9.|[2]Plosker GL. Pilsicainide. Drugs. 2010 Mar 5;70 (4) :455-67.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
Launched
Curated Selection
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