ERK-IN-2 (free base)
ERK-IN-2 free base is a ERK2 inhibitor with an IC50 value of 1.8 nM. ERK-IN-2 free base might lead to off-target toxicity and/or off-target activity at dose >10 μM[1].
Product Specifications
CAS Number
2743576-55-6
UNSPSC
12352005
Target
ERK
Type
Reference compound
Related Pathways
MAPK/ERK Pathway; Stem Cell/Wnt
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/erk-in-2-free-base.html
Solubility
10 mM in DMSO
Smiles
OCC1=C2C(NN=C2)=CC(NC(N[C@@H](C3=CC=CC=C3)C)=O)=N1
Molecular Formula
C16H17N5O2
Molecular Weight
311.34
References & Citations
[1]MRK-ERK Inhibitor and Negative Control.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
ERK2
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