Cavα2δ-IN-1
Cavα2δ-IN-1 shows high selectivity for voltage-gated calcium channels Cavα2δ-1 (Ki 6 nM) versus Cavα2δ-2 (Ki > 10000 nM) .
Product Specifications
CAS Number
2416957-09-8
UNSPSC
12352005
Target
Calcium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/cavα2δ-in-1.html
Solubility
10 mM in DMSO
Smiles
O=C1C(C=NC=C2)=C2N=C([C@H](N3C[C@@H](C)NCC3)CCC)N1CC
Molecular Formula
C18H27N5O
Molecular Weight
329.44
References & Citations
[1]Fernández A, et al. Piperazinyl Bicyclic Derivatives as Selective Ligands of the α2δ-1 Subunit of Voltage-Gated Calcium Channels. ACS Med Chem Lett. 2021 Oct 5;12 (11) :1802-1809.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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