CB2 receptor agonist 2

CB2 receptor agonist 2 is a potent and selective agonist for the CB2 (cannabinoid type 2) receptor with a Ki of 8.5 nM. CB2 receptor agonist 2 has high affinity and selectivity for CB2[1].

Product Specifications

CAS Number

[1314230-75-5]

UNSPSC

12352005

Target

Cannabinoid Receptor

Type

Reference compound

Related Pathways

GPCR/G Protein; Neuronal Signaling

Applications

Neuroscience-Neuromodulation

Field of Research

Neurological Disease

Assay Protocol

https://www.medchemexpress.com/cb2-receptor-agonist-2.html

Purity

99.9

Solubility

Ethanol : 30 mg/mL (ultrasonic; warming)

Smiles

O=C(C1=CN(CCCCC)C2=C(C1=O)C=C(C3=CC=CO3)C=C2OC)NC45CC6CC(C5)CC(C4)C6

Molecular Formula

C30H36N2O4

Molecular Weight

488.62

References & Citations

[1]Pasquini S, et al. Investigations on the 4-quinolone-3-carboxylic acid motif. 4. Identification of new potent and selective ligands for the cannabinoid type 2 receptor with diverse substitution patterns and antihyperalgesic effects in mice. J Med Chem. 2011;54 (15) :5444-5453.