GLP-1 receptor agonist 3
GLP-1 receptor agonist 3 (compound (R) -4A-1) is a GLP-1 receptor agonist (WO2018109607A1), used for diabetes research. compound (S) -4A-1 shows EC50s of 1.1 nM and 13 nM in Clone H6 and Clone C6 cell lines assay, respectively[1].
Product Specifications
CAS Number
2230200-09-4
UNSPSC
12352005
Target
GCGR
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Metabolism-sugar/lipid metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/glp-1-receptor-agonist-3.html
Solubility
10 mM in DMSO
Smiles
O=C(C1=CC=C2N=C(CN3CCC(C4=NC(OCC5=CC=C(C#N)C=C5F)=CC=C4)CC3)N(C[C@@H]6OCC6)C2=C1)O
Molecular Formula
C31H30FN5O4
Molecular Weight
555.60
References & Citations
[1]Gary Erik Aspnes, et al. Glp-1 receptor agonists and uses thereof. WO2018109607A1.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
LY420852 100 µg
PTPN20B (PTPN20) (NM_001042363) Human Over-expression Lysate
Sign In for Pricing
View Details 
100411F0-AAT 25 Tests
APC/iFluor® 700 Anti-human CD4 Antibody *RPA-T4*
Sign In for Pricing
View Details 