Apelin agonist 1
Apelin agonist 1 is an oral selective apelin agonist AM-2995, a agonist of the APJ (APLNR, angiotensin receptor like-1) receptor, may be used in the treatment of cardiovascular conditions. Apelin agonist 1 is extracted from patent WO 2018097944 (210.0), Example 210.0[1].
Product Specifications
CAS Number
2227512-85-6
UNSPSC
12352005
Target
Apelin Receptor (APJ)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/apelin-agonist-1.html
Solubility
10 mM in DMSO
Smiles
O=S(CCC1=CC=C(F)C=C1C#N)(NC2=NN=C(C3=CC=CO3)N2C4=C(OC)C=CC=C4OC)=O
Molecular Formula
C23H20FN5O5S
Molecular Weight
497.50
References & Citations
[1]Matthew Brown, et al. Triazole furan compounds as agonists of the apj receptor
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
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