Welcome to GenPrice! Check out our latest updates.

Shopping Cart (0)

Your cart is empty

Add some products to get started!

CK2-IN-9

CK2-IN-9 is a potent and selective inhibitor of CK2 kinase with an IC50 of 3 nM. CK2-IN-9 reduces Wnt reporter activity with an IC50 of 75 nM. CK2-IN-9 has low exposure (AUC=0.36 μM/h) and high clearance (CL=65 mL/min/kg) properties in rat[1].

Product Specifications

CAS Number

1461658-58-1

UNSPSC

12352005

Target

Casein Kinase; Wnt

Type

Reference compound

Related Pathways

Cell Cycle/DNA Damage; Stem Cell/Wnt

Applications

Cancer-Kinase/protease

Field of Research

Cancer

Assay Protocol

https://www.medchemexpress.com/ck2-in-9.html

Solubility

10 mM in DMSO

Smiles

O=C(C)NC1=CC(NC2=NC3=C(C#N)C=NN3C(NC4CC4)=C2)=CC=C1N(CCN(C)C)C

Molecular Formula

C23H29N9O

Molecular Weight

447.54

References & Citations

[1]Dowling JE, et al. Potent and Selective CK2 Kinase Inhibitors with Effects on Wnt Pathway Signaling in Vivo. ACS Med Chem Lett. 2016 Jan 20;7 (3) :300-5.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Frequently Asked Questions

More Discoveries

Explore Other Products

Browse additional items from our catalog

(2E) -3- (3-Chloro-1-benzothiophen-2-yl) prop-2-enoic acid
MJD76633-01 50 mg

(2E) -3- (3-Chloro-1-benzothiophen-2-yl) prop-2-enoic acid

Sign In for Pricing
View Details
(2E) -3- (3-Chloro-1-benzothiophen-2-yl) prop-2-enoic acid
MJD76633-02 0.5 g

(2E) -3- (3-Chloro-1-benzothiophen-2-yl) prop-2-enoic acid

Sign In for Pricing
View Details
Rat Fibroblast Growth Factor 11 (FGF11) CLIA Kit
MBS2709117-01 24 Strip Well

Rat Fibroblast Growth Factor 11 (FGF11) CLIA Kit

Sign In for Pricing
View Details
Rat Fibroblast Growth Factor 11 (FGF11) CLIA Kit
MBS2709117-02 48 Well

Rat Fibroblast Growth Factor 11 (FGF11) CLIA Kit

Sign In for Pricing
View Details
Rat Fibroblast Growth Factor 11 (FGF11) CLIA Kit
MBS2709117-03 96 Well

Rat Fibroblast Growth Factor 11 (FGF11) CLIA Kit

Sign In for Pricing
View Details
Rat Fibroblast Growth Factor 11 (FGF11) CLIA Kit
MBS2709117-04 5x 96 Well

Rat Fibroblast Growth Factor 11 (FGF11) CLIA Kit

Sign In for Pricing
View Details