CBK289001
CBK289001 is a tartrate-resistant acid phosphatase (TRAP/ACP5) inhibitor. CBK289001 inhibits TRAP 5bMV, TRAP 5bOX and TRAP 5aOX with IC50s of 125 μM, 4.21 μM and 14.2 μM, respectively[1].
Product Specifications
CAS Number
1212663-24-5
UNSPSC
12352005
Target
Protease Activated Receptor (PAR)
Type
Reference compound
Related Pathways
GPCR/G Protein
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/cbk289001.html
Purity
99.74
Solubility
DMSO : 100 mg/mL (ultrasonic)
Smiles
O=C(N1[C@H](C2=NC(C3=CC=C(OCO4)C4=C3)=NO2)CC5=C(NC=N5)C1)NC(C)C
Molecular Formula
C19H20N6O4
Molecular Weight
396.40
References & Citations
[1]Anja Reithmeier, et al. Identification of inhibitors of Tartrate-resistant acid phosphatase (TRAP/ACP5) activity by small-molecule screening. Chem Biol Drug Des. 2018 Jul;92 (1) :1255-1271.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Available Sizes
Frequently Asked Questions
More Discoveries
Explore Other Products
Browse additional items from our catalog
LC429100 20 µg
Matrilin 2 (MATN2) (NM_002380) Human Over-expression Lysate
Sign In for Pricing
View Details 
BNC471730-100 1x 100 µL
MMP3 (Marker of Metastasis and Rheumatoid Arthritis) (MMP3/1730), CF647 conjugate, 0.1mg/mL
Sign In for Pricing
View Details 
101001-2 1 mg
Spike S1 (B.1.1.7, Alpha Variant), Avi-His-Tag (SARS-CoV-2)
Sign In for Pricing
View Details 