3-Hydroxyphenazepam
3-Hydroxyphenazepam is an active metabolite of Cinazepam. Cinazepam is a GABAA receptor agonist. 3-Hydroxyphenazepam can inhibit synaptosomal transporter-mediated [3H]GABA uptake[1].
Product Specifications
CAS Number
70030-11-4
UNSPSC
12352005
Target
Drug Metabolite
Type
Reference compound
Related Pathways
Metabolic Enzyme/Protease
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/3-hydroxyphenazepam.html
Purity
99.90
Solubility
10 mM in DMSO
Smiles
BrC1=CC(C(C2=CC=CC=C2Cl)=NC3O)=C(C=C1)NC3=O
Molecular Formula
C15H10BrClN2O2
Molecular Weight
365.61
References & Citations
[1]Borisova T, et, al. GABAA receptor agonist cinazepam and its active metabolite 3-hydroxyphenazepam act differently at the presynaptic site. Eur Neuropsychopharmacol. 2021 Apr;45:39-51.
Shipping Conditions
Blue Ice
Storage Conditions
-20°C, 3 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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