GSK299115A
GSK299115A is a G Protein-coupled Receptor Kinase (GRK) and PKA inhibitor[1].
Product Specifications
CAS Number
[864082-35-9]
UNSPSC
12352005
Target
G Protein-coupled Receptor Kinase (GRK) ; PKA
Type
Reference compound
Related Pathways
GPCR/G Protein; Stem Cell/Wnt; TGF-beta/Smad
Applications
Cancer-Kinase/protease
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gsk299115a.html
Purity
98.99
Solubility
10 mM in DMSO
Smiles
O=C(NC1=CC2=C(C=C1)NN=C2)C3=C(NC(CC3C4=CC=C(C(Cl)=C4)Cl)=O)C
Molecular Formula
C20H16Cl2N4O2
Molecular Weight
415.27
References & Citations
[1]Homan KT, et al. Identification and structure-function analysis of subfamily selective G protein-coupled receptor kinase inhibitors. ACS Chem Biol. 2015 Jan 16;10 (1) :310-9.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
