Zolertine (hydrochloride)
Product Specifications
UNSPSC Description
Zolertine hydrochloride is an α-adrenoceptor antagonist with a pKi of 6.81 in rat liver (α1B-adrenoceptors) and 6.35 in rabbit liver (α1A-adrenoceptors) membranes[1].
Target Antigen
Adrenergic Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/zolertine-hydrochloride.html
Solubility
10 mM in DMSO
Smiles
[H]Cl.N1(CCN(CC1)CCC2=NN=NN2)C3=CC=CC=C3
Molecular Weight
294.78
References & Citations
[1]Ibarra M, et al. The alpha-adrenoceptor antagonist, zolertine, inhibits alpha1D- and alpha1A-adrenoceptor-mediated vasoconstriction in vitro. J Auton Pharmacol. 2000 Jun;20(3):139-45.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-123368/Zolertine-hydrochloride-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-123368/
Clinical Information
No Development Reported
CAS Number
7241-94-3
Curated Selection
Explore Other Products
Discover premium biology products from our extensive collection of 20M+ items
14954124 3 x 1.0μg DNA
CAMK1 CRISPRa sgRNA lentivector (set of three targets)(Mouse)
Ask
View Details