GR 128107
Product Specifications
UNSPSC Description
GR 128107 is a competitive melatonin receptor antagonist (pKi: 9.6)[1].
Target Antigen
Melatonin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein;Neuronal Signaling
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gr-128107.html
Solubility
10 mM in DMSO
Smiles
CC(N1CC(CCC1)C2=CNC3=C2C=C(C=C3)OC)=O
Molecular Weight
272.34
References & Citations
[1]Dubocovich ML, et al. Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor. Naunyn Schmiedebergs Arch Pharmacol. 1997 Mar;355(3):365-75.
Shipping Conditions
Room temperature
Product Datasheet
http://file.medchemexpress.com/batch_PDF/HY-120182/GR-128107-DataSheet-MedChemExpress.pdf
Product MSDS
http://file.medchemexpress.com/batch_PDF/HY-120182/
Clinical Information
No Development Reported
CAS Number
190328-44-0
Curated Selection
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