GR 128107
GR 128107 is a competitive melatonin receptor antagonist (pKi: 9.6) [1].
Product Specifications
CAS Number
[190328-44-0]
UNSPSC
12352005
Target
Melatonin Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/gr-128107.html
Solubility
10 mM in DMSO
Smiles
CC(N1CC(CCC1)C2=CNC3=C2C=C(C=C3)OC)=O
Molecular Formula
C16H20N2O2
Molecular Weight
272.34
References & Citations
[1]Dubocovich ML, et al. Melatonin receptor antagonists that differentiate between the human Mel1a and Mel1b recombinant subtypes are used to assess the pharmacological profile of the rabbit retina ML1 presynaptic heteroreceptor. Naunyn Schmiedebergs Arch Pharmacol. 1997 Mar;355 (3) :365-75.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Curated Selection
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