GSK215083
GSK215083 is a high affinity 5-HT6 receptor antagonist. GSK215083 can serves as a promising 5-HT6 radioligand candidate by radiolabeled with (11) C via methylation[1].
Product Specifications
CAS Number
607742-80-3
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/gsk215083.html
Solubility
10 mM in DMSO
Smiles
CN1CCN(CC1)C2=C3N=CC(S(=O)(C4=CC=CC(F)=C4)=O)=CC3=CC=C2
Molecular Formula
C20H20FN3O2S
Molecular Weight
385.46
References & Citations
[1]Parker CA, et al. Radiosynthesis and characterization of 11C-GSK215083 as a PET radioligand for the 5-HT6 receptor. J Nucl Med. 2012 Feb;53 (2) :295-303.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
5-HT6 Receptor; MUC2
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