RS-5773
RS-5773 is a calcium channel inhibitor and a diltiazem congener. RS-5773 has antianginal effect and does not cause excessive hypotension or depression of atrioventricular conduction [1].
Product Specifications
CAS Number
129173-57-5
UNSPSC
12352005
Target
Calcium Channel
Type
Reference compound
Related Pathways
Membrane Transporter/Ion Channel; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease; Cardiovascular Disease
Assay Protocol
https://www.medchemexpress.com/rs-5773.html
Solubility
10 mM in DMSO
Smiles
O=C1[C@@H]([C@@H](SC2=CC(CC3=CC=CS3)=CC=C2N1CCN(C)C)C4=CC=C(C=C4)OC)OC(C)=O.[H]Cl
Molecular Formula
C27H31ClN2O4S2
Molecular Weight
547.13
References & Citations
[1]H Shiga, et al. Antianginal effect of RS-5773, a diltiazem congener, in the methacholine-induced anginal model in rats. Jpn J Pharmacol . 1996 Dec;72 (4) :365-74.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
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