LY108742
LY108742 is a 5-HT2 receptor antagonist, with IC50 values of 9.3 nM (Rat), 57.2 nM (Pig), 56.8 nM (Monkey) [1].
Product Specifications
CAS Number
150196-69-3
UNSPSC
12352005
Target
5-HT Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/ly108742.html
Solubility
10 mM in DMSO
Smiles
O=C(OC(C)C(C)O)C(CC1C2=C3C4=CC=C2)CN(C1CC3=CN4C)C
Molecular Formula
C21H28N2O3
Molecular Weight
356.46
References & Citations
[1]D L Nelson, et al. Species differences in the pharmacology of the 5-hydroxytryptamine2 receptor: structurally specific differentiation by ergolines and tryptamines. J Pharmacol Exp Ther. 1993 Jun;265 (3) :1272-9.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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