FT001
FT001 is an orally active and selective BET inhibitor. FT001 has potent anti-proliferative effects against MV-4-11. FT001 can be used for research of cancer[1].
Product Specifications
CAS Number
[1778655-51-8]
UNSPSC
12352005
Target
Epigenetic Reader Domain
Type
Reference compound
Related Pathways
Epigenetics
Applications
Cancer-programmed cell death
Field of Research
Cancer
Assay Protocol
https://www.medchemexpress.com/ft001.html
Purity
99.90
Solubility
10 mM in DMSO
Smiles
O=C(C1CC1)N2C3=CC(C4=CC=C(N5CCS(=O)(CC5)=O)C=C4)=CC=C3N([C@H](C2)C)C(C)=O
Molecular Formula
C25H29N3O4S
Molecular Weight
467.58
References & Citations
[1]Millan DS, et al. Design and Optimization of Benzopiperazines as Potent Inhibitors of BET Bromodomains. ACS Med Chem Lett. 2017 Jul 14;8 (8) :847-852.
Shipping Conditions
Room Temperature
Storage Conditions
-20°C, 3 years; 4°C, 2 years (Powder)
Scientific Category
Reference compound1
Clinical Information
Phase 2
Available Sizes
Curated Selection
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