SR2595
SR2595 is an inverse agonist of PPARγ with an IC50 of 30 nM[1].
Product Specifications
CAS Number
1415252-61-7
UNSPSC
12352005
Target
PPAR
Type
Reference compound
Related Pathways
Cell Cycle/DNA Damage; Metabolic Enzyme/Protease; Vitamin D Related/Nuclear Receptor
Applications
Metabolism-protein/nucleotide metabolism
Field of Research
Metabolic Disease
Assay Protocol
https://www.medchemexpress.com/sr2595.html
Solubility
10 mM in DMSO
Smiles
CC(N1CC2=CC=C(C=C2)C3=CC=CC=C3C(O)=O)=C(C4=C1C=CC(C(N[C@H](C5=CC=C(C=C5)C(C)(C)C)C)=O)=C4)C
Molecular Formula
C37H38N2O3
Molecular Weight
558.71
References & Citations
[1]Marciano DP, et al. Pharmacological repression of PPARγ promotes osteogenesis. Nat Commun. 2015 Jun 12;6:7443.
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Isoform
PPARγ
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