LY2940094 (tartrate)
LY2940094 (BTRX-246040) tartrate is a potent, brain penetrant, selective and orally available N/OFQ peptide (NOP) receptor antagonist with high affinity (Ki=0.105 nM) and antagonist potency (Kb=0.166 nM) . LY2940094 tartrate reduces Ethanol self-administration and Ethanol seeking in animal models[1].
Product Specifications
CAS Number
[1307245-87-9]
Product Name Alternative
BTRX-246040 (tartrate)
UNSPSC
12352005
Hazard Statement
H302, H315, H319, H335
Target
Opioid Receptor
Type
Reference compound
Related Pathways
GPCR/G Protein; Neuronal Signaling
Applications
Neuroscience-Neuromodulation
Field of Research
Neurological Disease
Assay Protocol
https://www.medchemexpress.com/LY-2940094_tartrate.html
Concentration
10mM
Purity
99.66
Solubility
DMSO : 50 mg/mL (ultrasonic)
Smiles
OCC1=CC=CN=C1N2N=C(C)C(CN3CCC4(C5=C(C=C(Cl)S5)C(F)(F)CO4)CC3)=C2.O=C(O)[C@H](O)[C@@H](O)C(O)=O
Molecular Formula
C26H29ClF2N4O8S
Molecular Weight
631.05
Precautions
H302, H315, H319, H335
References & Citations
Shipping Conditions
Room Temperature
Storage Conditions
4°C (Powder, sealed storage, away from moisture)
Scientific Category
Reference compound1
Clinical Information
Phase 2
Isoform
NOP Receptor/ORL1
Available Sizes
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