VU0029767
VU0029767 is an allosteric enhancer of the M1 muscarinic receptor with the activity to modulate M1 receptor activity. VU0029767 can enhance M1 receptor activity by increasing agonist affinity, but exhibits different properties from other compounds under different experimental conditions, such as effects on mutant M1 receptors and effects on downstream signaling pathways.
Product Specifications
CAS Number
1134973-88-8
UNSPSC
12352005
Target
Others
Type
Reference compound
Related Pathways
Others
Field of Research
Others
Assay Protocol
https://www.medchemexpress.com/vu0029767.html
Smiles
O=C(N/N=C/C1=C2C=CC=CC2=CC=C1O)CNC3=CC=C(OCC)C=C3
Molecular Formula
C21H21N3O3
Molecular Weight
363.41
References & Citations
[1]Discovery and characterization of novel allosteric potentiators of M1 muscarinic receptors reveals multiple modes of activity
Shipping Conditions
Room temperature
Scientific Category
Reference compound1
Clinical Information
No Development Reported
Frequently Asked Questions
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