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PI3Kdelta inhibitor 1

PI3Kdelta inhibitor 1 (Compound 5d) is a potent, selective and orally available PI3Kδ inhibitor with an IC50 of 1.3 nM[1].

Product Specifications

CAS Number

[2242109-74-4]

UNSPSC

12352005

Target

PI3K

Type

Reference compound

Related Pathways

PI3K/Akt/mTOR

Applications

COVID-19-immunoregulation

Field of Research

Cancer; Inflammation/Immunology

Assay Protocol

https://www.medchemexpress.com/PI3Kdelta_inhibitor_1.html

Solubility

10 mM in DMSO

Smiles

CN1C2=NC(C3=CC(NS(C)(=O)=O)=C(OC)N=C3)=CC(OC[C@H]4CN(CCC5CCOCC5)CCC4)=C2C=N1

Molecular Formula

C27H38N6O5S

Molecular Weight

558.69

References & Citations

[1]Hamajima T, et al. Optimization and in vivo evaluation of pyrazolopyridines as a potent and selective PI3Kδ inhibitor. Bioorg Med Chem. 2018 Aug 7;26 (14) :3917-3924.

Shipping Conditions

Room temperature

Scientific Category

Reference compound1

Clinical Information

No Development Reported

Isoform

PI3Kδ

Curated Selection

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